Assay Detail
Binding
CHEMBL884570
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Inhibition constant against alpha adrenergic receptor
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 5 — Multiple protein complex / RNA |
| Curated By | Autocuration |
Publication
Designed multiple ligands. An emerging drug discovery paradigm.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 7.88 | 9.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL104229 | — | — | 1 | 9.00 |
| CHEMBL83617 | — | — | 1 | 7.80 |
| CHEMBL197982 | — | — | 1 | 6.85 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL104229 | — | Ki | = | 1.0 | nM | 9.00 |
| CHEMBL83617 | — | Ki | = | 16.0 | nM | 7.80 |
| CHEMBL197982 | — | Ki | = | 140.0 | nM | 6.85 |