Assay Detail
Binding
CHEMBL884756
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Inhibitory activity against Mandelate racemase at pH 7.5 at 25 degree C
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Pseudomonas putida |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Inhibition of mandelate racemase by the substrate-intermediate-product analogue 1,1-diphenyl-1-hydroxymethylphosphonate.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 5.33 | 5.33 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL24720 | ALPHA HYDROXY BENZYLPHOSPHONATE | — | 1 | 5.33 |
| CHEMBL1161801 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL24720 | ALPHA HYDROXY BENZYLPHOSPHONATE | Ki | = | 4700.0 | nM | 5.33 |
| CHEMBL1161801 | — | Ki | = | 1410000.0 | nM | - |