Assay Detail
Binding
CHEMBL885189
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibitory concentration against acetylcholinesterase
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Designed multiple ligands. An emerging drug discovery paradigm.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 7.43 | 7.85 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL197696 | — | — | 1 | 7.85 |
| CHEMBL194372 | — | — | 1 | 7.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL197696 | — | IC50 | = | 14.0 | nM | 7.85 |
| CHEMBL194372 | — | IC50 | = | 101.0 | nM | 7.00 |