Assay Detail
Binding
CHEMBL889722
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of human FGFR1 kinase expressed in insect cell by HTRF detection method
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Novel inhibitor for fibroblast growth factor receptor tyrosine kinase.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 6.16 | 6.40 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL231526 | — | — | 1 | 6.40 |
| CHEMBL358728 | — | — | 1 | 5.92 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL231526 | — | IC50 | = | 400.0 | nM | 6.40 |
| CHEMBL358728 | — | IC50 | = | 1200.0 | nM | 5.92 |