Assay Detail
ADMET
CHEMBL890920
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Cytotoxicity against J774.1 cells after 48 hrs
11
Total Activities
11
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | ADMET |
| Organism | Mus musculus |
| Cell Type | J774.1 |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Antitrypanosomal activity of quaternary naphthalimide derivatives.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 11 | 5.49 | 5.49 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL388891 | — | — | 1 | 5.49 |
| CHEMBL233476 | — | — | 1 | - |
| CHEMBL8532 | — | — | 1 | - |
| CHEMBL269592 | — | — | 1 | - |
| CHEMBL397958 | — | — | 1 | - |
| CHEMBL388470 | — | — | 1 | - |
| CHEMBL390702 | — | — | 1 | - |
| CHEMBL233049 | — | — | 1 | - |
| CHEMBL406691 | — | — | 1 | - |
| CHEMBL8449 | — | — | 1 | - |
| CHEMBL389344 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL388891 | — | IC50 | = | 3240.0 | nM | 5.49 |
| CHEMBL233476 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL8532 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL269592 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL397958 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL388470 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL390702 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL233049 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL406691 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL8449 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL389344 | — | IC50 | > | 100000.0 | nM | - |