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Assay Detail

CHEMBL896872

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity to PR
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Intermediate

Target

Progesterone receptor (CHEMBL208)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Substituted 6-(1-pyrrolidine)quinolin-2(1H)-ones as novel selective androgen receptor modulators.
Martinborough E, Shen Y, Oeveren Av, Long YO, Lau TL, Marschke KB, Chang WY, López FJ, Vajda EG, Rix PJ, Viveros OH, Negro-Vilar A, Zhi L.
J Med Chem (2007) 50 : 5049 -5052
PubMed 17887661 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 5.60 5.60

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL467888 LGD-2941 1.0 1 5.60

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL467888 LGD-2941 Ki = 2500.0 nM 5.60