Assay Detail
Functional
CHEMBL898609
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antagonist activity at ERalpha expressed in yeast AH109 assessed as inhibition of 17-beta-estradiol induced alpha-galactosidase activity
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Intermediate |
Publication
Aza analogues of equol: novel ligands for estrogen receptor beta.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.42 | 5.58 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL391619 | — | — | 1 | 5.58 |
| CHEMBL392029 | — | — | 1 | 5.25 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL391619 | — | IC50 | = | 2650.0 | nM | 5.58 |
| CHEMBL392029 | — | IC50 | = | 5570.0 | nM | 5.25 |