Assay Detail
Binding
CHEMBL902327
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Displacement of human [125I]PYY from NPY2 receptor expressed in human KAN-TS cells
17
Total Activities
17
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | KAN-TS |
| Confidence | 9 — Direct single protein target |
| Curated By | Intermediate |
Publication
Identification of selective neuropeptide Y2 peptide agonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 17 | 7.83 | 9.40 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL439904 | — | — | 1 | 9.40 |
| CHEMBL238533 | — | — | 1 | 8.52 |
| CHEMBL241105 | — | — | 1 | 8.40 |
| CHEMBL227456 | — | — | 1 | 8.40 |
| CHEMBL411765 | — | — | 1 | 8.30 |
| CHEMBL397528 | — | — | 1 | 8.22 |
| CHEMBL437290 | — | — | 1 | 8.22 |
| CHEMBL436630 | — | — | 1 | 8.22 |
| CHEMBL266814 | — | — | 1 | 8.22 |
| CHEMBL269267 | — | — | 1 | 8.05 |
| CHEMBL411766 | — | — | 1 | 7.75 |
| CHEMBL392889 | — | — | 1 | 7.52 |
| CHEMBL411793 | — | — | 1 | 7.12 |
| CHEMBL429005 | — | — | 1 | 7.02 |
| CHEMBL397529 | — | — | 1 | 6.96 |
| CHEMBL268200 | — | — | 1 | 6.57 |
| CHEMBL397527 | — | — | 1 | 6.17 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL439904 | — | Ki | = | 0.4 | nM | 9.40 |
| CHEMBL238533 | — | Ki | = | 3.0 | nM | 8.52 |
| CHEMBL241105 | — | Ki | = | 4.0 | nM | 8.40 |
| CHEMBL227456 | — | Ki | = | 4.0 | nM | 8.40 |
| CHEMBL411765 | — | Ki | = | 5.0 | nM | 8.30 |
| CHEMBL397528 | — | Ki | = | 6.0 | nM | 8.22 |
| CHEMBL437290 | — | Ki | = | 6.0 | nM | 8.22 |
| CHEMBL436630 | — | Ki | = | 6.0 | nM | 8.22 |
| CHEMBL266814 | — | Ki | = | 6.0 | nM | 8.22 |
| CHEMBL269267 | — | Ki | = | 9.0 | nM | 8.05 |
| CHEMBL411766 | — | Ki | = | 18.0 | nM | 7.75 |
| CHEMBL392889 | — | Ki | = | 30.0 | nM | 7.52 |
| CHEMBL411793 | — | Ki | = | 75.0 | nM | 7.12 |
| CHEMBL429005 | — | Ki | = | 95.0 | nM | 7.02 |
| CHEMBL397529 | — | Ki | = | 110.0 | nM | 6.96 |
| CHEMBL268200 | — | Ki | = | 270.0 | nM | 6.57 |
| CHEMBL397527 | — | Ki | = | 670.0 | nM | 6.17 |