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Assay Detail

CHEMBL906759

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Functional
Nitric oxide scavenging activity assessed as inhibition of DAF2 oxidation
8
Total Activities
8
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

2-Styrylchromones: novel strong scavengers of reactive oxygen and nitrogen species.
Gomes A, Fernandes E, Silva AM, Santos CM, Pinto DC, Cavaleiro JA, Lima JL.
Bioorg Med Chem (2007) 15 : 6027 -6036
PubMed 17624791 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 8 5.85 6.62

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL228623 1 6.62
CHEMBL374371 1 6.54
CHEMBL374372 1 6.47
CHEMBL228622 1 6.29
CHEMBL50 QUERCETIN 3.0 1 5.71
CHEMBL151 LUTEOLIN 2.0 1 5.58
CHEMBL226335 RUTIN 3.0 1 5.44
CHEMBL415858 1 4.13

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL228623 IC50 = 240.0 nM 6.62
CHEMBL374371 IC50 = 290.0 nM 6.54
CHEMBL374372 IC50 = 340.0 nM 6.47
CHEMBL228622 IC50 = 510.0 nM 6.29
CHEMBL50 QUERCETIN IC50 = 1950.0 nM 5.71
CHEMBL151 LUTEOLIN IC50 = 2610.0 nM 5.58
CHEMBL226335 RUTIN IC50 = 3660.0 nM 5.44
CHEMBL415858 IC50 = 73900.0 nM 4.13