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Assay Detail

CHEMBL910469

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antibacterial activity against Escherichia coli K12 by broth microdilution method
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Escherichia coli
Confidence 1 — Organism
Curated By Intermediate

Target

Escherichia coli (CHEMBL354)
Type ORGANISM
Organism Escherichia coli

Publication

Isoprenoid biosynthesis as a drug target: bisphosphonate inhibition of Escherichia coli K12 growth and synergistic effects of fosmidomycin.
Leon A, Liu L, Yang Y, Hudock MP, Hall P, Yin F, Studer D, Puan KJ, Morita CT, Oldfield E.
J Med Chem (2006) 49 : 7331 -7341
PubMed 17149863 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 5.57 6.66

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL203125 FOSMIDOMYCIN 3.0 1 6.66
CHEMBL56073 1 4.48

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL203125 FOSMIDOMYCIN IC50 = 220.0 nM 6.66
CHEMBL56073 IC50 = 33000.0 nM 4.48