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Assay Detail

CHEMBL910791

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of Plasmodium falciparum ENR by fluorescence quenching in presence of ECG
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Plasmodium falciparum
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Enoyl-acyl-carrier protein reductase (CHEMBL4150)
Type SINGLE PROTEIN
Organism Plasmodium falciparum

Publication

Green tea catechins potentiate triclosan binding to enoyl-ACP reductase from Plasmodium falciparum (PfENR).
Sharma SK, Parasuraman P, Kumar G, Surolia N, Surolia A.
J Med Chem (2007) 50 : 765 -775
PubMed 17263522 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 7.55 7.55

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL849 TRICLOSAN 4.0 1 7.55

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL849 TRICLOSAN Ki = 28.31 nM 7.55