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Assay Detail

CHEMBL916716

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Displacement of 3H]RX821002 from rat cortex adrenergic alpha-2 receptor
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Rattus norvegicus
Confidence 5 — Multiple protein complex / RNA
Curated By Autocuration

Target

Adrenergic receptor alpha-2 (CHEMBL2093864)
Type PROTEIN FAMILY
Organism Rattus norvegicus

Publication

Novel sigma receptor ligands: synthesis and biological profile.
Prezzavento O, Campisi A, Ronsisvalle S, Li Volti G, Marrazzo A, Bramanti V, Cannavò G, Vanella L, Cagnotto A, Mennini T, Ientile R, Ronsisvalle G.
J Med Chem (2007) 50 : 951 -961
PubMed 17328523 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 5.03 5.03

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL222301 1 5.03

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL222301 Ki = 9414.0 nM 5.03