Assay Detail
Functional
CHEMBL917185
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Agonistic activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically evoked twitch
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Mus musculus |
| Tissue | Vas deferens |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Highly selective fluorescent analogue of the potent delta-opioid receptor antagonist Dmt-Tic.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 8.59 | 8.59 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2369958 | — | — | 1 | 8.59 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2369958 | — | IC50 | = | 2.58 | nM | 8.59 |