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Assay Detail

CHEMBL918106

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Binding
Inhibition of Escherichia coli TEM1
8
Total Activities
8
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Escherichia coli
Confidence 9 — Direct single protein target
Curated By Intermediate

Target

Beta-lactamase TEM (CHEMBL2065)
Type SINGLE PROTEIN
Organism Escherichia coli

Publication

Structure-activity relationship of 6-methylidene penems bearing tricyclic heterocycles as broad-spectrum beta-lactamase inhibitors: crystallographic structures show unexpected binding of 1,4-thiazepine intermediates.
Venkatesan AM, Gu Y, Dos Santos O, Abe T, Agarwal A, Yang Y, Petersen PJ, Weiss WJ, Mansour TS, Nukaga M, Hujer AM, Bonomo RA, Knox JR.
J Med Chem (2004) 47 : 6556 -6568
PubMed 15588091 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 8 8.08 9.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL122450 1 9.00
CHEMBL222375 1 8.52
CHEMBL388778 1 8.22
CHEMBL222922 1 8.10
CHEMBL222866 1 8.05
CHEMBL222758 1 8.00
CHEMBL375172 1 7.75
CHEMBL1439 TAZOBACTAM SODIUM 4.0 1 7.00

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL122450 IC50 = 1.0 nM 9.00
CHEMBL222375 IC50 = 3.0 nM 8.52
CHEMBL388778 IC50 = 6.0 nM 8.22
CHEMBL222922 IC50 = 8.0 nM 8.10
CHEMBL222866 IC50 = 9.0 nM 8.05
CHEMBL222758 IC50 = 10.0 nM 8.00
CHEMBL375172 IC50 = 18.0 nM 7.75
CHEMBL1439 TAZOBACTAM SODIUM IC50 = 100.0 nM 7.00