Assay Detail
Functional
CHEMBL920122
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Inhibition of IL5 in mouse Y16 cells at 50 uM
27
Total Activities
27
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Mus musculus |
| Cell Type | Y16 |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Structural requirement of chalcones for the inhibitory activity of interleukin-5.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 27 | 4.94 | 5.75 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL374181 | — | — | 1 | 5.75 |
| CHEMBL224931 | — | — | 1 | 5.41 |
| CHEMBL224163 | — | — | 1 | 5.35 |
| CHEMBL224055 | — | — | 1 | 5.19 |
| CHEMBL375693 | — | — | 1 | 5.19 |
| CHEMBL225094 | — | — | 1 | 5.16 |
| CHEMBL375893 | — | — | 1 | 5.15 |
| CHEMBL224577 | — | — | 1 | 5.03 |
| CHEMBL390327 | — | — | 1 | 4.99 |
| CHEMBL225402 | — | — | 1 | 4.97 |
| CHEMBL225129 | — | — | 1 | 4.90 |
| CHEMBL390095 | — | — | 1 | 4.85 |
| CHEMBL224294 | — | — | 1 | 4.85 |
| CHEMBL224890 | — | — | 1 | 4.84 |
| CHEMBL224539 | — | — | 1 | 4.67 |
| CHEMBL225401 | — | — | 1 | 4.60 |
| CHEMBL1370 | BUDESONIDE | 4.0 | 1 | 4.57 |
| CHEMBL224054 | — | — | 1 | 4.55 |
| CHEMBL388403 | — | — | 1 | 4.54 |
| CHEMBL126804 | — | — | 1 | 4.32 |
| CHEMBL224407 | — | — | 1 | - |
| CHEMBL224833 | — | — | 1 | - |
| CHEMBL224753 | — | — | 1 | - |
| CHEMBL425122 | — | — | 1 | - |
| CHEMBL225353 | — | — | 1 | - |
| CHEMBL437678 | — | — | 1 | - |
| CHEMBL224480 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL374181 | — | IC50 | = | 1800.0 | nM | 5.75 |
| CHEMBL224931 | — | IC50 | = | 3900.0 | nM | 5.41 |
| CHEMBL224163 | — | IC50 | = | 4500.0 | nM | 5.35 |
| CHEMBL224055 | — | IC50 | = | 6400.0 | nM | 5.19 |
| CHEMBL375693 | — | IC50 | = | 6400.0 | nM | 5.19 |
| CHEMBL225094 | — | IC50 | = | 7000.0 | nM | 5.16 |
| CHEMBL375893 | — | IC50 | = | 7100.0 | nM | 5.15 |
| CHEMBL224577 | — | IC50 | = | 9400.0 | nM | 5.03 |
| CHEMBL390327 | — | IC50 | = | 10200.0 | nM | 4.99 |
| CHEMBL225402 | — | IC50 | = | 10800.0 | nM | 4.97 |
| CHEMBL225129 | — | IC50 | = | 12600.0 | nM | 4.90 |
| CHEMBL390095 | — | IC50 | = | 14200.0 | nM | 4.85 |
| CHEMBL224294 | — | IC50 | = | 14100.0 | nM | 4.85 |
| CHEMBL224890 | — | IC50 | = | 14300.0 | nM | 4.84 |
| CHEMBL224539 | — | IC50 | = | 21400.0 | nM | 4.67 |
| CHEMBL225401 | — | IC50 | = | 25300.0 | nM | 4.60 |
| CHEMBL1370 | BUDESONIDE | IC50 | = | 26800.0 | nM | 4.57 |
| CHEMBL224054 | — | IC50 | = | 27900.0 | nM | 4.55 |
| CHEMBL388403 | — | IC50 | = | 28800.0 | nM | 4.54 |
| CHEMBL126804 | — | IC50 | = | 48200.0 | nM | 4.32 |
| CHEMBL224407 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL224833 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL224753 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL425122 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL225353 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL437678 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL224480 | — | IC50 | > | 50000.0 | nM | - |