Assay Detail

CHEMBL924524

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Functional

Agonist activity at rat beta-3 adrenergic receptor

ChEMBL ↗

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Target

Beta-3 adrenergic receptor (CHEMBL4031) ↗

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Primary target Beta-3 adrenergic receptor

CHEMBL4031

Anchored from Assay target.

Protein identity Beta-3 adrenergic receptor

Disease frame Disease evidence pending

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Review focus Open DB context pending

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Total Activities

Compounds Tested

Activity Types

Assay Parameters

Assay Information

Assay Type	Functional
Organism	Rattus norvegicus
Confidence	9 — Direct single protein target
Curated By	Intermediate

Target

Beta-3 adrenergic receptor (CHEMBL4031) ↗

Type	SINGLE PROTEIN
Organism	Rattus norvegicus

Publication

Potent oxindole based human beta3 adrenergic receptor agonists.

Stevens FC, Bloomquist WE, Borel AG, Cohen ML, Droste CA, Heiman ML, Kriauciunas A, Sall DJ, Tinsley FC, Jesudason CD.
Bioorg Med Chem Lett (2007) 17 : 6270 -6273
PubMed 17911024 · DOI

Activity Statistics

Type	Count	Avg pChEMBL	Best pChEMBL
EC50	1	8.19	8.19

Compounds Tested

Compound	Name	Phase	Activities	Best pChEMBL
CHEMBL251372	—	—	1	8.19

Activity Data

Compound	Name	Type	Rel.	Value	Units	pChEMBL
CHEMBL251372	—	EC50	=	6.5	nM	8.19