Assay Detail
Binding
CHEMBL925174
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Inhibition of rat OSC
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Confidence | 9 — Direct single protein target |
| Curated By | Intermediate |
Publication
The biology and chemistry of hyperlipidemia.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 4 | 7.02 | 7.30 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL253784 | — | — | 1 | 7.30 |
| CHEMBL64905 | — | — | 1 | 7.30 |
| CHEMBL253785 | — | — | 1 | 7.30 |
| CHEMBL253787 | — | — | 1 | 6.16 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL253784 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL64905 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL253785 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL253787 | — | IC50 | = | 700.0 | nM | 6.16 |