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Assay Detail

CHEMBL927607

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Binding
Inhibition of bovine PNMT by radiochemical assay
14
Total Activities
14
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Bos taurus
Confidence 9 — Direct single protein target
Curated By Intermediate

Target

Phenylethanolamine N-methyltransferase (CHEMBL2331)
Type SINGLE PROTEIN
Organism Bos taurus

Publication

Synthesis of 4,5,6,7-tetrahydrothieno[3,2-c]pyridines and comparison with their isosteric 1,2,3,4-tetrahydroisoquinolines as inhibitors of phenylethanolamine N-methyltransferase.
Grunewald GL, Seim MR, Bhat SR, Wilson ME, Criscione KR.
Bioorg Med Chem (2008) 16 : 542 -559
PubMed 18024134 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 14 6.30 8.51

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL287837 1 8.51
CHEMBL281864 1 7.25
CHEMBL357424 1 7.17
CHEMBL59719 1 7.14
CHEMBL281289 1 6.92
CHEMBL26717 1 6.55
CHEMBL60434 1 5.85
CHEMBL27162 1 5.82
CHEMBL26711 1 5.70
CHEMBL14346 1,2,3,4-TETRAHYDROISOQUINOLINE 1 5.30
CHEMBL26879 1 5.30
CHEMBL28228 1 4.14
CHEMBL610 PHENETHYLAMINE 1 -
CHEMBL522 BENZYLAMINE 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL287837 Ki = 3.1 nM 8.51
CHEMBL281864 Ki = 56.0 nM 7.25
CHEMBL357424 Ki = 67.0 nM 7.17
CHEMBL59719 Ki = 72.0 nM 7.14
CHEMBL281289 Ki = 120.0 nM 6.92
CHEMBL26717 Ki = 280.0 nM 6.55
CHEMBL60434 Ki = 1400.0 nM 5.85
CHEMBL27162 Ki = 1500.0 nM 5.82
CHEMBL26711 Ki = 2000.0 nM 5.70
CHEMBL14346 1,2,3,4-TETRAHYDROISOQUINOLINE Ki = 5000.0 nM 5.30
CHEMBL26879 Ki = 5000.0 nM 5.30
CHEMBL28228 Ki = 72000.0 nM 4.14
CHEMBL610 PHENETHYLAMINE Ki = 220000.0 nM -
CHEMBL522 BENZYLAMINE Ki = 170000.0 nM -