Assay Detail
ADMET
CHEMBL933670
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Antiproliferative activity against BMDM cells
9
Total Activities
9
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | ADMET |
| Cell Type | BMDM |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Structure-based optimization of a potent class of arylamide FMS inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 9 | 8.22 | 9.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL257154 | — | — | 1 | 9.00 |
| CHEMBL252436 | — | — | 1 | 8.70 |
| CHEMBL254702 | — | — | 1 | 8.70 |
| CHEMBL402337 | — | — | 1 | 8.44 |
| CHEMBL256712 | — | — | 1 | 8.10 |
| CHEMBL256950 | — | — | 1 | 7.52 |
| CHEMBL429855 | — | — | 1 | 7.10 |
| CHEMBL258238 | — | — | 1 | - |
| CHEMBL257153 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL257154 | — | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL252436 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL254702 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL402337 | — | IC50 | = | 3.6 | nM | 8.44 |
| CHEMBL256712 | — | IC50 | = | 8.0 | nM | 8.10 |
| CHEMBL256950 | — | IC50 | = | 30.0 | nM | 7.52 |
| CHEMBL429855 | — | IC50 | = | 80.0 | nM | 7.10 |
| CHEMBL258238 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL257153 | — | IC50 | > | 1000.0 | nM | - |