Assay Detail
Functional
CHEMBL935038
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antiviral activity against HCV assessed as inhibition of HCV RNA replication in OR6 cells after 72 hrs by luciferase reporter assay
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Hepacivirus hominis |
| Cell Type | OR6 |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
Comprehensive analysis of the effects of ordinary nutrients on hepatitis C virus RNA replication in cell culture.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 6 | 4.81 | 5.42 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1536 | ERGOCALCIFEROL | 4.0 | 1 | 5.42 |
| CHEMBL1293 | BETA CAROTENE | 4.0 | 1 | 5.20 |
| CHEMBL267476 | LINOLEIC ACID | 2.0 | 1 | 4.70 |
| CHEMBL15594 | ARACHIDONIC ACID | -1.0 | 1 | 4.66 |
| CHEMBL460026 | ICOSAPENT | 3.0 | 1 | 4.44 |
| CHEMBL367149 | DOCONEXENT | 3.0 | 1 | 4.43 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1536 | ERGOCALCIFEROL | EC50 | = | 3800.0 | nM | 5.42 |
| CHEMBL1293 | BETA CAROTENE | EC50 | = | 6300.0 | nM | 5.20 |
| CHEMBL267476 | LINOLEIC ACID | EC50 | = | 20200.0 | nM | 4.70 |
| CHEMBL15594 | ARACHIDONIC ACID | EC50 | = | 22100.0 | nM | 4.66 |
| CHEMBL460026 | ICOSAPENT | EC50 | = | 36200.0 | nM | 4.44 |
| CHEMBL367149 | DOCONEXENT | EC50 | = | 37000.0 | nM | 4.43 |