Assay Detail
Binding
CHEMBL937670
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Inhibition of FGFR1
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
A systematic interaction map of validated kinase inhibitors with Ser/Thr kinases.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 6.58 | 7.67 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL189584 | PD-173074 | — | 1 | 7.67 |
| CHEMBL13485 | SU-11652 | — | 1 | 6.77 |
| CHEMBL86943 | — | — | 1 | 5.30 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL189584 | PD-173074 | IC50 | = | 21.5 | nM | 7.67 |
| CHEMBL13485 | SU-11652 | IC50 | = | 170.0 | nM | 6.77 |
| CHEMBL86943 | — | IC50 | = | 5000.0 | nM | 5.30 |