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Assay Detail

CHEMBL938421

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against Herpes simplex virus 1 F infected in african green monkey Vero cells assessed as plaque reduction after 36 to 48 hrs
11
Total Activities
11
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Human alphaherpesvirus 1
Cell Type Vero
Confidence 1 — Organism
Curated By Intermediate

Target

Human alphaherpesvirus 1 (CHEMBL377)
Type ORGANISM
Organism Human alphaherpesvirus 1

Publication

Sensitivity of monkey B virus (Cercopithecine herpesvirus 1) to antiviral drugs: role of thymidine kinase in antiviral activities of substrate analogs and acyclonucleosides.
Focher F, Lossani A, Verri A, Spadari S, Maioli A, Gambino JJ, Wright GE, Eberle R, Black DH, Medveczky P, Medveczky M, Shugar D.
Antimicrob Agents Chemother (2007) 51 : 2028 -2034
PubMed 17438061 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 11 5.69 6.92

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL31634 BRIVUDINE 2.0 1 6.92
CHEMBL182 GANCICLOVIR 4.0 1 6.16
CHEMBL184 ACYCLOVIR 4.0 1 5.85
CHEMBL318153 EDOXUDINE 2.0 1 5.68
CHEMBL788 IDOXURIDINE 4.0 1 5.55
CHEMBL1540 PENCICLOVIR 4.0 1 5.33
CHEMBL1090 VIDARABINE 4.0 1 5.16
CHEMBL5314375 CIDOFOVIR 4.0 1 4.84
CHEMBL666 FOSCARNET 4.0 1 -
CHEMBL406254 1 -
CHEMBL1129 TRIFLURIDINE 4.0 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL31634 BRIVUDINE EC50 = 120.0 nM 6.92
CHEMBL182 GANCICLOVIR EC50 = 700.0 nM 6.16
CHEMBL184 ACYCLOVIR EC50 = 1400.0 nM 5.85
CHEMBL318153 EDOXUDINE EC50 = 2100.0 nM 5.68
CHEMBL788 IDOXURIDINE EC50 = 2800.0 nM 5.55
CHEMBL1540 PENCICLOVIR EC50 = 4700.0 nM 5.33
CHEMBL1090 VIDARABINE EC50 = 7000.0 nM 5.16
CHEMBL5314375 CIDOFOVIR EC50 = 14400.0 nM 4.84
CHEMBL666 FOSCARNET EC50 = 250000.0 nM -
CHEMBL406254 EC50 = 330000.0 nM -
CHEMBL1129 TRIFLURIDINE EC50 < 1700.0 nM -