Assay Detail
Binding
CHEMBL938652
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of FAAH in rat brain assessed as hydrolysis of anandamide
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Tissue | Brain |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Discovery and development of fatty acid amide hydrolase (FAAH) inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 6.10 | 6.10 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL6206 | BROMOENOL LACTONE | — | 1 | 6.10 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL6206 | BROMOENOL LACTONE | IC50 | = | 800.0 | nM | 6.10 |