Assay Detail
Binding
CHEMBL939372
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Inhibition of Src
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Expert |
Target
Proto-oncogene tyrosine-protein kinase Src (CHEMBL267) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
A systematic interaction map of validated kinase inhibitors with Ser/Thr kinases.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 7 | 6.09 | 6.55 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL605003 | — | — | 1 | 6.55 |
| CHEMBL260138 | ALSTERPAULLONE 2 | — | 1 | 6.50 |
| CHEMBL1276317 | — | — | 1 | 6.37 |
| CHEMBL258726 | — | — | 1 | 5.66 |
| CHEMBL437612 | — | — | 1 | 5.36 |
| CHEMBL406375 | — | — | 1 | - |
| CHEMBL261238 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL605003 | — | IC50 | = | 280.0 | nM | 6.55 |
| CHEMBL260138 | ALSTERPAULLONE 2 | IC50 | = | 316.23 | nM | 6.50 |
| CHEMBL1276317 | — | IC50 | = | 430.0 | nM | 6.37 |
| CHEMBL258726 | — | IC50 | = | 2200.0 | nM | 5.66 |
| CHEMBL437612 | — | IC50 | = | 4400.0 | nM | 5.36 |
| CHEMBL406375 | — | IC50 | >= | 10000.0 | nM | - |
| CHEMBL261238 | — | IC50 | > | 400000000.0 | nM | - |