Assay Detail
Binding
CHEMBL944037
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Inhibition of MMP9
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Intermediate |
Publication
A novel series of highly selective inhibitors of MMP-3.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 5.51 | 6.39 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL398641 | — | — | 1 | 6.39 |
| CHEMBL251917 | — | — | 1 | 5.62 |
| CHEMBL250266 | — | — | 1 | 4.52 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL398641 | — | IC50 | = | 406.0 | nM | 6.39 |
| CHEMBL251917 | — | IC50 | = | 2420.0 | nM | 5.62 |
| CHEMBL250266 | — | IC50 | = | 30400.0 | nM | 4.52 |