Assay Detail
Binding
CHEMBL946607
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [3H]estradiol from human recombinant ERalpha
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Isolation and structure elucidation of an isoflavone and a sesterterpenoic acid from Henriettella fascicularis.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 5.43 | 6.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL44 | GENISTEIN | 2.0 | 1 | 6.52 |
| CHEMBL512579 | — | — | 1 | 4.99 |
| CHEMBL8145 | DAIDZEIN | 2.0 | 1 | 4.77 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL44 | GENISTEIN | IC50 | = | 300.0 | nM | 6.52 |
| CHEMBL512579 | — | IC50 | = | 10200.0 | nM | 4.99 |
| CHEMBL8145 | DAIDZEIN | IC50 | = | 17000.0 | nM | 4.77 |