Assay Detail
Binding
CHEMBL947530
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Inhibition of protein phosphatase 2A
8
Total Activities
8
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
The 1990 United States-Japan seminar on bioorganic marine chemistry, meeting report.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 8 | 9.05 | 9.05 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL430266 | CALYCULIN A | — | 1 | 9.05 |
| CHEMBL443660 | CALYCULIN D | — | 1 | 9.05 |
| CHEMBL509059 | CALYCULIN | — | 1 | 9.05 |
| CHEMBL487898 | CALYCULIN B | — | 1 | 9.05 |
| CHEMBL510956 | CALYCULIN H | — | 1 | 9.05 |
| CHEMBL489660 | CALYCULIN G | — | 1 | 9.05 |
| CHEMBL452909 | CALYCULIN F | — | 1 | 9.05 |
| CHEMBL446220 | CALYCULIN E | — | 1 | 9.05 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL430266 | CALYCULIN A | IC50 | = | 0.9 | nM | 9.05 |
| CHEMBL443660 | CALYCULIN D | IC50 | = | 0.9 | nM | 9.05 |
| CHEMBL509059 | CALYCULIN | IC50 | = | 0.9 | nM | 9.05 |
| CHEMBL487898 | CALYCULIN B | IC50 | = | 0.9 | nM | 9.05 |
| CHEMBL510956 | CALYCULIN H | IC50 | = | 0.9 | nM | 9.05 |
| CHEMBL489660 | CALYCULIN G | IC50 | = | 0.9 | nM | 9.05 |
| CHEMBL452909 | CALYCULIN F | IC50 | = | 0.9 | nM | 9.05 |
| CHEMBL446220 | CALYCULIN E | IC50 | = | 0.9 | nM | 9.05 |