Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL947576

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of COX1
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Intermediate

Target

Prostaglandin G/H synthase 1 (CHEMBL221)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Two new stilbene dimer glucosides from grape (Vitis vinifera) cell cultures.
Waffo-Teguo P, Lee D, Cuendet M, Mérillon J, Pezzuto JM, Kinghorn AD.
J Nat Prod (2001) 64 : 136 -138
PubMed 11170689 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 3 4.98 5.37

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL518935 1 5.37
CHEMBL503412 1 5.28
CHEMBL480462 PALLIDOL 1 4.30

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL518935 IC50 = 4300.0 nM 5.37
CHEMBL503412 IC50 = 5200.0 nM 5.28
CHEMBL480462 PALLIDOL IC50 = 50000.0 nM 4.30