Assay Detail
Binding
CHEMBL948074
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Binding affinity to 5HT2A receptor
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Total synthesis and evaluation of [18F]MHMZ.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 9.57 | 9.89 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL62919 | ALTANSERIN | 2.0 | 1 | 9.89 |
| CHEMBL74355 | VOLINANSERIN | 3.0 | 1 | 9.24 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL62919 | ALTANSERIN | Ki | = | 0.13 | nM | 9.89 |
| CHEMBL74355 | VOLINANSERIN | Ki | = | 0.57 | nM | 9.24 |