Assay Detail
Functional
CHEMBL952125
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Suppression of TNFalpha production in LPS-stimulated whole blood
21
Total Activities
21
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Tissue | Blood |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Discovery of kinase inhibitors by high-throughput docking and scoring based on a transferable linear interaction energy model.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 21 | 8.39 | 9.15 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL327959 | — | — | 1 | 9.15 |
| CHEMBL327746 | — | — | 1 | 9.15 |
| CHEMBL328614 | — | — | 1 | 9.00 |
| CHEMBL319556 | — | — | 1 | 8.89 |
| CHEMBL97227 | — | — | 1 | 8.85 |
| CHEMBL94825 | — | — | 1 | 8.80 |
| CHEMBL96763 | — | — | 1 | 8.70 |
| CHEMBL96487 | — | — | 1 | 8.54 |
| CHEMBL96225 | — | — | 1 | 8.42 |
| CHEMBL96345 | — | — | 1 | 8.40 |
| CHEMBL327987 | — | — | 1 | 8.36 |
| CHEMBL96432 | — | — | 1 | 8.35 |
| CHEMBL328242 | — | — | 1 | 8.25 |
| CHEMBL271528 | — | — | 1 | 8.15 |
| CHEMBL271750 | — | — | 1 | 8.12 |
| CHEMBL94417 | — | — | 1 | 8.11 |
| CHEMBL316604 | — | — | 1 | 8.00 |
| CHEMBL94444 | — | — | 1 | 7.94 |
| CHEMBL419140 | — | — | 1 | 7.91 |
| CHEMBL270956 | — | — | 1 | 7.57 |
| CHEMBL327217 | — | — | 1 | 7.57 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL327959 | — | IC50 | = | 0.7 | nM | 9.15 |
| CHEMBL327746 | — | IC50 | = | 0.7 | nM | 9.15 |
| CHEMBL328614 | — | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL319556 | — | IC50 | = | 1.3 | nM | 8.89 |
| CHEMBL97227 | — | IC50 | = | 1.4 | nM | 8.85 |
| CHEMBL94825 | — | IC50 | = | 1.6 | nM | 8.80 |
| CHEMBL96763 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL96487 | — | IC50 | = | 2.9 | nM | 8.54 |
| CHEMBL96225 | — | IC50 | = | 3.8 | nM | 8.42 |
| CHEMBL96345 | — | IC50 | = | 4.0 | nM | 8.40 |
| CHEMBL327987 | — | IC50 | = | 4.4 | nM | 8.36 |
| CHEMBL96432 | — | IC50 | = | 4.5 | nM | 8.35 |
| CHEMBL328242 | — | IC50 | = | 5.6 | nM | 8.25 |
| CHEMBL271528 | — | IC50 | = | 7.0 | nM | 8.15 |
| CHEMBL271750 | — | IC50 | = | 7.6 | nM | 8.12 |
| CHEMBL94417 | — | IC50 | = | 7.8 | nM | 8.11 |
| CHEMBL316604 | — | IC50 | = | 10.1 | nM | 8.00 |
| CHEMBL94444 | — | IC50 | = | 11.4 | nM | 7.94 |
| CHEMBL419140 | — | IC50 | = | 12.2 | nM | 7.91 |
| CHEMBL270956 | — | IC50 | = | 27.1 | nM | 7.57 |
| CHEMBL327217 | — | IC50 | = | 26.8 | nM | 7.57 |