Assay Detail
Binding
CHEMBL952691
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Binding affinity to beta-1 adrenoceptor
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Intermediate |
Publication
Antagonists of the calcium receptor I. Amino alcohol-based parathyroid hormone secretagogues.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 4 | 8.52 | 8.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL486278 | — | — | 1 | 8.52 |
| CHEMBL2112075 | — | — | 1 | - |
| CHEMBL504479 | — | — | 1 | - |
| CHEMBL523475 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL486278 | — | EC50 | = | 3.0 | nM | 8.52 |
| CHEMBL2112075 | — | EC50 | - | — | - | |
| CHEMBL504479 | — | EC50 | - | — | - | |
| CHEMBL523475 | — | EC50 | - | — | - |