Assay Detail
Binding
CHEMBL956561
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [3H]CP-55940 from CB1 receptor in mouse brain at 100 nM
2
Total Activities
1
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Mus musculus |
| Tissue | Brain |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Monoacylglycerol lipase regulates 2-arachidonoylglycerol action and arachidonic acid levels.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 1 | 9.07 | 9.07 |
| Bmax | 1 | - | - |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL444970 | CHLORPHRIFOS OXON | — | 2 | 9.07 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL444970 | CHLORPHRIFOS OXON | Kd | = | 0.86 | nM | 9.07 |
| CHEMBL444970 | CHLORPHRIFOS OXON | Bmax | = | 0.17 | pmol/mg | - |