Assay Detail
ADMET
CHEMBL957933
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Antiproliferative activity against mouse J774.A1 cells after 72 hrs by MTT conversion assay
13
Total Activities
13
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | ADMET |
| Organism | Mus musculus |
| Cell Type | J774.A1 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Antiproliferative oleanane saponins from Meryta denhamii.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 13 | 5.99 | 8.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1425 | MERCAPTOPURINE ANHYDROUS | 4.0 | 1 | 8.52 |
| CHEMBL486881 | — | — | 1 | 6.72 |
| CHEMBL507138 | — | — | 1 | 6.50 |
| CHEMBL506188 | — | — | 1 | 5.60 |
| CHEMBL449916 | — | — | 1 | 5.52 |
| CHEMBL499677 | — | — | 1 | 5.44 |
| CHEMBL507155 | — | — | 1 | 5.41 |
| CHEMBL502666 | — | — | 1 | 5.16 |
| CHEMBL524337 | — | — | 1 | 5.05 |
| CHEMBL509910 | — | — | 1 | - |
| CHEMBL452712 | — | — | 1 | - |
| CHEMBL505247 | — | — | 1 | - |
| CHEMBL448367 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1425 | MERCAPTOPURINE ANHYDROUS | IC50 | = | 3.0 | nM | 8.52 |
| CHEMBL486881 | — | IC50 | = | 190.0 | nM | 6.72 |
| CHEMBL507138 | — | IC50 | = | 320.0 | nM | 6.50 |
| CHEMBL506188 | — | IC50 | = | 2500.0 | nM | 5.60 |
| CHEMBL449916 | — | IC50 | = | 3000.0 | nM | 5.52 |
| CHEMBL499677 | — | IC50 | = | 3600.0 | nM | 5.44 |
| CHEMBL507155 | — | IC50 | = | 3900.0 | nM | 5.41 |
| CHEMBL502666 | — | IC50 | = | 6900.0 | nM | 5.16 |
| CHEMBL524337 | — | IC50 | = | 9000.0 | nM | 5.05 |
| CHEMBL509910 | — | IC50 | - | — | - | |
| CHEMBL452712 | — | IC50 | - | — | - | |
| CHEMBL505247 | — | IC50 | - | — | - | |
| CHEMBL448367 | — | IC50 | - | — | - |