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Assay Detail

CHEMBL962074

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antioxidant activity assessed as inhibition of lactoperoxidase-catalyzed oxidation of 2,2'-azinobis(3-ethylbenzthione 6-sulfonic acid)
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Confidence 1 — Organism
Curated By Autocuration

Publication

Interaction of methimazole with I2: X-ray crystal structure of the charge transfer complex methimazole-I2. implications for the mechanism of action of methimazole-based antithyroid drugs.
Isaia F, Aragoni MC, Arca M, Demartin F, Devillanova FA, Floris G, Garau A, Hursthouse MB, Lippolis V, Medda R, Oppo F, Pira M, Verani G.
J Med Chem (2008) 51 : 4050 -4053
PubMed 18529045 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 5.55 5.85

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL452810 1 5.85
CHEMBL1515 METHIMAZOLE 4.0 1 5.25

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL452810 IC50 = 1400.0 nM 5.85
CHEMBL1515 METHIMAZOLE IC50 = 5600.0 nM 5.25