Assay Detail
Binding
CHEMBL962376
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Inhibition of His6x-tagged Plasmodium falciparum PfPK5 expressed in Escherichia coli by microtiter plate scintillation counting
19
Total Activities
19
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Plasmodium falciparum |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Selective inhibition of Pfmrk, a Plasmodium falciparum CDK, by antimalarial 1,3-diaryl-2-propenones.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 19 | 4.00 | 4.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL446640 | — | — | 1 | 4.00 |
| CHEMBL470424 | — | — | 1 | - |
| CHEMBL16947 | WR-190433 | — | 1 | - |
| CHEMBL506696 | — | — | 1 | - |
| CHEMBL221741 | — | — | 1 | - |
| CHEMBL139856 | — | — | 1 | - |
| CHEMBL221432 | — | — | 1 | - |
| CHEMBL385631 | — | — | 1 | - |
| CHEMBL218330 | — | — | 1 | - |
| CHEMBL450678 | — | — | 1 | - |
| CHEMBL509932 | — | — | 1 | - |
| CHEMBL187682 | — | — | 1 | - |
| CHEMBL471252 | — | — | 1 | - |
| CHEMBL471253 | — | — | 1 | - |
| CHEMBL471254 | — | — | 1 | - |
| CHEMBL471667 | — | — | 1 | - |
| CHEMBL187926 | — | — | 1 | - |
| CHEMBL468255 | — | — | 1 | - |
| CHEMBL511497 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL446640 | — | IC50 | = | 100000.0 | nM | 4.00 |
| CHEMBL470424 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL16947 | WR-190433 | IC50 | > | 382000.0 | nM | - |
| CHEMBL506696 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL221741 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL139856 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL221432 | — | IC50 | - | — | - | |
| CHEMBL385631 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL218330 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL450678 | — | IC50 | > | 360000.0 | nM | - |
| CHEMBL509932 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL187682 | — | IC50 | > | 316000.0 | nM | - |
| CHEMBL471252 | — | IC50 | > | 315000.0 | nM | - |
| CHEMBL471253 | — | IC50 | > | 268000.0 | nM | - |
| CHEMBL471254 | — | IC50 | > | 256000.0 | nM | - |
| CHEMBL471667 | — | IC50 | = | 123000.0 | nM | - |
| CHEMBL187926 | — | IC50 | > | 302000.0 | nM | - |
| CHEMBL468255 | — | IC50 | > | 299000.0 | nM | - |
| CHEMBL511497 | — | IC50 | > | 100000.0 | nM | - |