Assay Detail
Binding
CHEMBL964244
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of FGFR1K autophosphorylation activity assessed as [32P] incorporation
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Intermediate |
Publication
Structures of the tyrosine kinase domain of fibroblast growth factor receptor in complex with inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.00 | 5.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL315546 | — | — | 1 | 5.00 |
| CHEMBL89363 | — | — | 1 | 5.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL315546 | — | IC50 | = | 10000.0 | nM | 5.00 |
| CHEMBL89363 | — | IC50 | = | 10000.0 | nM | 5.00 |