Assay Detail
Binding
CHEMBL965323
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Inhibition of DPP8
26
Total Activities
26
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Intermediate |
Publication
Discovery of new binding elements in DPP-4 inhibition and their applications in novel DPP-4 inhibitor design.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 26 | 4.54 | 5.68 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL433572 | — | — | 1 | 5.68 |
| CHEMBL510073 | — | — | 1 | 4.82 |
| CHEMBL512887 | — | — | 1 | 4.77 |
| CHEMBL527424 | — | — | 1 | 4.75 |
| CHEMBL488484 | — | — | 1 | 4.57 |
| CHEMBL452297 | — | — | 1 | 4.57 |
| CHEMBL452290 | — | — | 1 | 4.41 |
| CHEMBL507738 | — | — | 1 | 4.39 |
| CHEMBL488678 | — | — | 1 | 4.37 |
| CHEMBL488637 | — | — | 1 | 4.33 |
| CHEMBL471936 | — | — | 1 | 4.19 |
| CHEMBL388475 | — | — | 1 | 4.12 |
| CHEMBL452805 | — | — | 1 | 4.06 |
| CHEMBL452289 | — | — | 1 | - |
| CHEMBL512895 | — | — | 1 | - |
| CHEMBL472123 | — | — | 1 | - |
| CHEMBL442673 | — | — | 1 | - |
| CHEMBL472124 | — | — | 1 | - |
| CHEMBL504506 | — | — | 1 | - |
| CHEMBL527198 | — | — | 1 | - |
| CHEMBL488469 | — | — | 1 | - |
| CHEMBL519591 | — | — | 1 | - |
| CHEMBL487630 | — | — | 1 | - |
| CHEMBL520067 | — | — | 1 | - |
| CHEMBL220249 | — | — | 1 | - |
| CHEMBL507719 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL433572 | — | IC50 | = | 2100.0 | nM | 5.68 |
| CHEMBL510073 | — | IC50 | = | 15000.0 | nM | 4.82 |
| CHEMBL512887 | — | IC50 | = | 17000.0 | nM | 4.77 |
| CHEMBL527424 | — | IC50 | = | 18000.0 | nM | 4.75 |
| CHEMBL488484 | — | IC50 | = | 27000.0 | nM | 4.57 |
| CHEMBL452297 | — | IC50 | = | 27000.0 | nM | 4.57 |
| CHEMBL452290 | — | IC50 | = | 39000.0 | nM | 4.41 |
| CHEMBL507738 | — | IC50 | = | 41000.0 | nM | 4.39 |
| CHEMBL488678 | — | IC50 | = | 43000.0 | nM | 4.37 |
| CHEMBL488637 | — | IC50 | = | 47000.0 | nM | 4.33 |
| CHEMBL471936 | — | IC50 | = | 64000.0 | nM | 4.19 |
| CHEMBL388475 | — | IC50 | = | 75000.0 | nM | 4.12 |
| CHEMBL452805 | — | IC50 | = | 87000.0 | nM | 4.06 |
| CHEMBL452289 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL512895 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL472123 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL442673 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL472124 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL504506 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL527198 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL488469 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL519591 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL487630 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL520067 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL220249 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL507719 | — | IC50 | > | 100000.0 | nM | - |