Assay Detail
Functional
CHEMBL972303
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of collagen-induced platelet aggregation in human blood after 3 mins by turbidimetric assay
54
Total Activities
54
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Tissue | Blood |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Synthesis and anti-platelet evaluation of 2-benzoylaminobenzoate analogs.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 54 | 4.16 | 4.31 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL468147 | — | — | 1 | 4.31 |
| CHEMBL451176 | — | — | 1 | 4.11 |
| CHEMBL513337 | — | — | 1 | 4.06 |
| CHEMBL452104 | — | — | 1 | - |
| CHEMBL467785 | — | — | 1 | - |
| CHEMBL6 | INDOMETHACIN | 4.0 | 1 | - |
| CHEMBL249828 | — | — | 1 | - |
| CHEMBL401138 | — | — | 1 | - |
| CHEMBL249829 | — | — | 1 | - |
| CHEMBL250467 | — | — | 1 | - |
| CHEMBL399683 | — | — | 1 | - |
| CHEMBL250468 | — | — | 1 | - |
| CHEMBL250469 | — | — | 1 | - |
| CHEMBL250654 | — | — | 1 | - |
| CHEMBL430020 | — | — | 1 | - |
| CHEMBL399844 | — | — | 1 | - |
| CHEMBL467764 | — | — | 1 | - |
| CHEMBL506055 | — | — | 1 | - |
| CHEMBL513179 | — | — | 1 | - |
| CHEMBL468956 | — | — | 1 | - |
| CHEMBL467777 | — | — | 1 | - |
| CHEMBL468957 | — | — | 1 | - |
| CHEMBL467950 | — | — | 1 | - |
| CHEMBL468148 | — | — | 1 | - |
| CHEMBL512115 | — | — | 1 | - |
| CHEMBL468770 | — | — | 1 | - |
| CHEMBL468771 | — | — | 1 | - |
| CHEMBL466355 | — | — | 1 | - |
| CHEMBL467955 | — | — | 1 | - |
| CHEMBL467778 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL468147 | — | IC50 | = | 48800.0 | nM | 4.31 |
| CHEMBL451176 | — | IC50 | = | 77000.0 | nM | 4.11 |
| CHEMBL513337 | — | IC50 | = | 87800.0 | nM | 4.06 |
| CHEMBL6 | INDOMETHACIN | IC50 | > | 100000.0 | nM | - |
| CHEMBL468814 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL467785 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL452104 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL498361 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL497551 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL498997 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL495682 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL498777 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL498776 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL525561 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL468153 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL468152 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL467801 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL467800 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL467956 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL467784 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL468023 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL467783 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL513825 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL469156 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL468996 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL447195 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL513179 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL467778 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL467955 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL466355 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL468771 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL468770 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL512115 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL468148 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL467950 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL468957 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL467777 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL468956 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL249828 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL506055 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL467764 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL399844 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL430020 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL250654 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL250469 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL250468 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL399683 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL250467 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL249829 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL401138 | — | IC50 | > | 100000.0 | nM | - |