Assay Detail
Binding
CHEMBL976623
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of Crotalus adamanteus venom phospholipase A2 by fluorometric assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Crotalus adamanteus |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Hyrtiazepine, an azepino-indole-type alkaloid from the Red Sea marine sponge Hyrtios erectus.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.63 | 6.40 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL463914 | MANOALIDE | — | 1 | 6.40 |
| CHEMBL465767 | HYRTIOSULAWESINE | — | 1 | 4.85 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL463914 | MANOALIDE | IC50 | = | 400.0 | nM | 6.40 |
| CHEMBL465767 | HYRTIOSULAWESINE | IC50 | = | 14000.0 | nM | 4.85 |