Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL983166

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Inhibition of LPS-induced nitric oxide production in mouse RAW264.7 cells by Griess method
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Mus musculus
Cell Type RAW264.7
Confidence 1 — Organism
Curated By Autocuration

Target

RAW264.7 (CHEMBL612557)
Type CELL-LINE
Organism Mus musculus

Publication

Saponins from Cussonia bancoensis and their inhibitory effects on nitric oxide production.
Tapondjou LA, Lontsi D, Sondengam BL, Shaheen F, Choudhary MI, Atta-ur-Rahman, van Heerden FR, Park HJ, Lee KT.
J Nat Prod (2003) 66 : 1266 -1269
PubMed 14510614 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 5 4.72 5.58

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL523622 1 5.58
CHEMBL7889 L-NIL 1 4.73
CHEMBL461104 1 4.66
CHEMBL169 URSOLIC ACID 2.0 1 4.33
CHEMBL506997 1 4.32

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL523622 IC50 = 2600.0 nM 5.58
CHEMBL7889 L-NIL IC50 = 18600.0 nM 4.73
CHEMBL461104 IC50 = 22100.0 nM 4.66
CHEMBL169 URSOLIC ACID IC50 = 46900.0 nM 4.33
CHEMBL506997 IC50 = 47900.0 nM 4.32