Assay Detail
Functional
CHEMBL990222
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antiinflammatory activity in human PMNC assessed as inhibition of proliferation
8
Total Activities
8
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Monoterpene glycosides and triterpene acids from Eriobotrya deflexa.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 8 | 5.06 | 7.92 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL160 | CYCLOSPORINE | 4.0 | 1 | 7.92 |
| CHEMBL518162 | — | — | 1 | 4.57 |
| CHEMBL239075 | EUSCAPHIC ACID | — | 1 | 4.54 |
| CHEMBL461068 | — | — | 1 | 4.49 |
| CHEMBL461703 | — | — | 1 | 4.42 |
| CHEMBL459413 | — | — | 1 | 4.40 |
| CHEMBL459616 | — | — | 1 | - |
| CHEMBL515705 | ARJUNIC ACID | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL160 | CYCLOSPORINE | IC50 | = | 12.0 | nM | 7.92 |
| CHEMBL518162 | — | IC50 | = | 26900.0 | nM | 4.57 |
| CHEMBL239075 | EUSCAPHIC ACID | IC50 | = | 28800.0 | nM | 4.54 |
| CHEMBL461068 | — | IC50 | = | 32500.0 | nM | 4.49 |
| CHEMBL461703 | — | IC50 | = | 38100.0 | nM | 4.42 |
| CHEMBL459413 | — | IC50 | = | 40000.0 | nM | 4.40 |
| CHEMBL459616 | — | IC50 | - | — | - | |
| CHEMBL515705 | ARJUNIC ACID | IC50 | - | — | - |