Assay Detail
Binding
CHEMBL990573
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Displacement of [3H]CCPA from rat adenosine A1 receptor
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Synthesis and adenosine receptor binding studies of some novel triazolothienopyrimidines.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 4 | 6.57 | 9.30 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL183 | 1,3-DIPROPYL-8-CYCLOPENTYLXANTHINE [DPCPX] | — | 1 | 9.30 |
| CHEMBL522879 | — | — | 1 | 5.93 |
| CHEMBL453690 | — | — | 1 | 5.68 |
| CHEMBL510505 | — | — | 1 | 5.36 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL183 | 1,3-DIPROPYL-8-CYCLOPENTYLXANTHINE [DPCPX] | Ki | = | 0.5 | nM | 9.30 |
| CHEMBL522879 | — | Ki | = | 1170.0 | nM | 5.93 |
| CHEMBL453690 | — | Ki | = | 2100.0 | nM | 5.68 |
| CHEMBL510505 | — | Ki | = | 4400.0 | nM | 5.36 |