Assay Detail
Functional
CHEMBL991620
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Cytotoxicity against cisplatin-resistant human C13 cells after 48 hrs
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | C13 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Identification of novel protein kinase CK1 delta (CK1delta) inhibitors through structure-based virtual screening.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 4.58 | 5.10 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL88326 | — | — | 1 | 5.10 |
| CHEMBL86771 | — | — | 1 | 4.06 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL88326 | — | IC50 | = | 8000.0 | nM | 5.10 |
| CHEMBL86771 | — | IC50 | = | 87900.0 | nM | 4.06 |