Assay Detail
Binding
CHEMBL992671
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [3H]diprenorphine from mouse delta opioid receptor expressed in CHO cells
8
Total Activities
8
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Mus musculus |
| Cell Type | CHO |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Synthesis and biological evaluation of C-12 triazole and oxadiazole analogs of salvinorin A.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 8 | 8.54 | 8.54 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL140050 | ETORPHINE | 2.0 | 1 | 8.54 |
| CHEMBL210564 | — | — | 1 | - |
| CHEMBL475987 | — | — | 1 | - |
| CHEMBL514358 | — | — | 1 | - |
| CHEMBL474275 | — | — | 1 | - |
| CHEMBL474477 | — | — | 1 | - |
| CHEMBL478509 | — | — | 1 | - |
| CHEMBL478139 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL140050 | ETORPHINE | Ki | = | 2.9 | nM | 8.54 |
| CHEMBL210564 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL475987 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL514358 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL474275 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL474477 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL478509 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL478139 | — | Ki | > | 1000.0 | nM | - |