Assay Detail
Functional
CHEMBL998017
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Agonist activity at androgen receptor
15
Total Activities
15
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Confidence | 8 — Homologous single protein target |
| Curated By | Intermediate |
Publication
Nonsteroidal selective androgen receptor modulators (SARMs): dissociating the anabolic and androgenic activities of the androgen receptor for therapeutic benefit.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 15 | 8.52 | 9.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL296323 | — | — | 1 | 9.52 |
| CHEMBL233773 | — | — | 1 | 9.35 |
| CHEMBL229861 | — | — | 1 | 9.05 |
| CHEMBL467790 | — | — | 1 | 8.96 |
| CHEMBL436784 | — | — | 1 | 8.82 |
| CHEMBL467888 | LGD-2941 | 1.0 | 1 | 8.82 |
| CHEMBL333745 | — | — | 1 | 8.78 |
| CHEMBL512283 | — | — | 1 | 8.77 |
| CHEMBL229264 | — | — | 1 | 8.68 |
| CHEMBL125236 | — | — | 1 | 8.40 |
| CHEMBL3084525 | — | — | 1 | 8.30 |
| CHEMBL124718 | — | — | 1 | 8.21 |
| CHEMBL224263 | — | — | 1 | 8.15 |
| CHEMBL467887 | — | — | 1 | 7.83 |
| CHEMBL242469 | — | — | 1 | 6.20 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL296323 | — | Ki | = | 0.3 | nM | 9.52 |
| CHEMBL233773 | — | Ki | = | 0.45 | nM | 9.35 |
| CHEMBL229861 | — | Ki | = | 0.9 | nM | 9.05 |
| CHEMBL467790 | — | Ki | = | 1.1 | nM | 8.96 |
| CHEMBL436784 | — | Ki | = | 1.5 | nM | 8.82 |
| CHEMBL467888 | LGD-2941 | Ki | = | 1.5 | nM | 8.82 |
| CHEMBL333745 | — | Ki | = | 1.65 | nM | 8.78 |
| CHEMBL512283 | — | Ki | = | 1.7 | nM | 8.77 |
| CHEMBL229264 | — | Ki | = | 2.1 | nM | 8.68 |
| CHEMBL125236 | — | Ki | = | 4.0 | nM | 8.40 |
| CHEMBL3084525 | — | Ki | = | 5.0 | nM | 8.30 |
| CHEMBL124718 | — | Ki | = | 6.1 | nM | 8.21 |
| CHEMBL224263 | — | Ki | = | 7.1 | nM | 8.15 |
| CHEMBL467887 | — | Ki | = | 14.9 | nM | 7.83 |
| CHEMBL242469 | — | Ki | = | 630.0 | nM | 6.20 |