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Compound Detail

CHEMBL1096215

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CCCCCCCCC(=O)O[C@]12[C@H]([C@@H]3C=C(CO)C[C@]4(O)C(=O)C(C)=C[C@H]4[C@@]3(O)C[C@H]1OC(=O)c1ccccc1)C2(C)C

Basic Information

ChEMBL ID CHEMBL1096215
Phase Preclinical
Structure Type MOL
InChI Key XCZMBPWIQJRZDE-VSHBPWGQSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

594.8
MW (Da)
4.85
ALogP
8
HBA
3
HBD
130.4
PSA (Ų)
0.19
QED
1
Ro5 Violations
11
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C35H46O8
MW 594.75
Aromatic Rings 1
Heavy Atoms 43
NP-Likeness 2.21

Activity Summary

IC50 1 meas. best 8.0

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
RAW264.7
CHEMBL612557
IC50 8.0 8.0 10.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
RAW264.7 IC50 = 10.0 nM 8.0 Antiinflammatory activity against mouse RAW264.7 cells assessed as inhibition of... 20192236

Literature References

PubMed DOI Target Context # Activities
20192236 10.1021/np9005053 RAW264.7 1

Data from ChEMBL 36 via Core Engine