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Compound Detail

CHEMBL114648

BETA-NAPHTOIC ACID
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O=C(O)c1ccc2ccccc2c1

Basic Information

ChEMBL ID CHEMBL114648
Name BETA-NAPHTOIC ACID
Phase Preclinical
Structure Type MOL
InChI Key UOBYKYZJUGYBDK-UHFFFAOYSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
12
Publications
0
Known Names

Molecular Properties

172.2
MW (Da)
2.54
ALogP
1
HBA
1
HBD
37.3
PSA (Ų)
0.72
QED
0
Ro5 Violations
1
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C11H8O2
MW 172.18
Aromatic Rings 2
Heavy Atoms 13
NP-Likeness -0.18

Activity Summary

IC50 1 meas. best 4.21

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
IC50 4.21 4.21 61400.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Unchecked IC50 = 61400.0 nM 4.21 Antagonist activity at Gloeobacter violaceus ligand-gated ion channel expressed ... 23682762

Literature References

PubMed DOI Target Context # Activities
23682762 10.1021/jm400374q Unchecked 2
24499135 10.1021/jm401808n Staphylococcus aureus 2
671456 10.1021/jm00204a015 Rattus norvegicus 2
1527790 10.1021/jm00096a014 No relevant target 1
1527790 10.1021/jm00096a014 ADMET 1
3820229 10.1021/jm00386a022 Polyunsaturated fatty acid 5-lipoxygenase 1
23136941 10.1021/jf3038874 Meloidogyne incognita 1
23682762 10.1021/jm400374q No relevant target 1
24249037 10.1007/s11095-013-1232-z No relevant target 1
24499135 10.1021/jm401808n Quinolone resistance protein NorA 1
915902 10.1021/jm00221a013 Unchecked 1
26154240 10.1016/j.bmc.2015.06.042 Curvularia lunata 1

Data from ChEMBL 36 via Core Engine