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Compound Detail

CHEMBL1170269

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COC(=O)c1cc(C(=O)OC)cc(-c2ccc(O[C@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@@H]3O)cc2)c1

Basic Information

ChEMBL ID CHEMBL1170269
Phase Preclinical
Structure Type MOL
InChI Key AJLVSCOTDPQPFW-FNIAAEIWSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
2
Publications
0
Known Names

Molecular Properties

448.4
MW (Da)
0.11
ALogP
10
HBA
4
HBD
152.0
PSA (Ų)
0.45
QED
0
Ro5 Violations
6
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C22H24O10
MW 448.42
Aromatic Rings 2
Heavy Atoms 32
NP-Likeness 0.87

Activity Summary

EC50 1 meas. best 7.11

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
EC50 7.11 7.11 77.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Unchecked EC50 = 77.0 nM 7.11 Displacement of 5(6)-FAM-mannoside from Escherichia coli FimH by fluorescence po... 20507142

Literature References

PubMed DOI Target Context # Activities
20507142 10.1021/jm100438s Unchecked 3
22449031 10.1021/jm300165m Unchecked 2

Data from ChEMBL 36 via Core Engine