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Compound Detail

CHEMBL1200728

GUANIDINE HYDROCHLORIDE
💊 Approved Drug
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💊 Approved Drug

Basic Information

ChEMBL ID CHEMBL1200728
Name GUANIDINE HYDROCHLORIDE
Phase Approved
Structure Type MOL
InChI Key PJJJBBJSCAKJQF-UHFFFAOYSA-N
Therapeutic ✓ Yes
Parent Compound CHEMBL821
Active Moiety CHEMBL821

Known Names

Guanidine hydrochloride NSC-755884
0
Targets
13
Activities
3
Assay Types
0
PK Parameters
9
Publications
2
Known Names
3
Indications
1
Mechanisms

Molecular Properties

59.1
MW (Da)
-1.16
ALogP
1
HBA
3
HBD
75.9
PSA (Ų)
0.24
QED
0
Ro5 Violations
0
Rot. Bonds

Drug Information

Molecule Type Small molecule
First Approval 1939
Availability Discontinued
Chirality Achiral

Routes of Administration

Oral
USAN Stem guan-

Extended Properties

Molecular Formula CH6ClN3
MW 95.53
Aromatic Rings 0
Heavy Atoms 4
NP-Likeness 0.32

Mechanism of Action

Mechanism Action Type Target Direct Efficacy
Voltage-gated potassium channel blocker BLOCKER Voltage-gated potassium channel

Indications

Carcinoma, Small Cell Lambert-Eaton Myasthenic Syndrome Muscle Weakness

Activity Summary

EC50 7 meas.
IC50 5 meas.
Ki 1 meas.

Literature References

PubMed DOI Target Context # Activities
32250117 10.1021/acs.jmedchem.9b01955 L-lactate dehydrogenase B chain 18
31881489 10.1016/j.ejmech.2019.112007 Coxsackievirus B3 5
31447248 10.1016/j.bmc.2019.115052 Complement C5 4
20014752 10.1021/tx900326k Hepatotoxicity 3
- 10.6019/CHEMBL4495565 SARS-CoV-2 2
25466178 10.1016/j.bmcl.2014.11.004 Nucleic Acid 1
- 10.21203/rs.3.rs-23951/v1 SARS-CoV-2 1
- 10.6019/CHEMBL4495564 Replicase polyprotein 1ab 1
36063653 10.1016/j.bmc.2022.116970 Unchecked 1

Data from ChEMBL 36 via Core Engine