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Compound Detail

CHEMBL1236642

VACCENIC ACID
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CCCCCC/C=C\CCCCCCCCCC(=O)O

Basic Information

ChEMBL ID CHEMBL1236642
Name VACCENIC ACID
Phase Preclinical
Structure Type MOL
InChI Key UWHZIFQPPBDJPM-FPLPWBNLSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
2
Publications
0
Known Names

Molecular Properties

282.5
MW (Da)
6.11
ALogP
1
HBA
1
HBD
37.3
PSA (Ų)
0.29
QED
1
Ro5 Violations
15
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C18H34O2
MW 282.47
Aromatic Rings 0
Heavy Atoms 20
NP-Likeness 0.87

Activity Summary

IC50 1 meas. best 4.8

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Telomerase reverse transcriptase
CHEMBL2916
IC50 4.8 4.8 16000.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Telomerase reverse transcriptase IC50 = 16000.0 nM 4.8 Inhibition of telomerase extracted from human K562 cells preincubated for 10 min... -

Literature References

PubMed DOI Target Context # Activities
- 10.1039/C0MD00241K Telomerase reverse transcriptase 1
28704049 10.1021/acs.jnatprod.6b00823 Albumin 1

Data from ChEMBL 36 via Core Engine